SCHEMBL9192192

SCHEMBL9192192

O=c1[nH]c(CSCc2ccccc2)nc2nccnc12

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
ALDH1A1 P00352 1/20 0.45
CYP2C19 P33261 1/20 0.45
HCAR2 Q8TDS4 6/20 0.45
PIK3C2A O00443 1/20 0.43
TP53 P04637 1/20 0.40
PLA2G7 Q13093 2/20 0.38
MAOB P27338 1/20 0.38
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 1/20 0.38
DAO P14920 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27248301 0.80 TP53 (0.60) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL9189988 0.78 HCAR2 (0.56) RAB9AHCAR2
SCHEMBL9195100 0.75 RAB9A (0.59) NPC1RAB9ASMN1; SMN2HCAR2TP53
SCHEMBL3817859 0.71 TNKS2 (0.44) SMN1; SMN2ALDH1A1HCAR2TP53
SCHEMBL1624031 0.71 TNKS (0.50) SMN1; SMN2HCAR2
SCHEMBL9501020 0.71 HCAR2 (0.33) ALDH1A1HCAR2KMT2A
SCHEMBL1624717 0.70 HCAR2 (0.55) HCAR2PLA2G7DAO
SCHEMBL9191917 0.69 ADORA2A (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1CYP2C19
SCHEMBL9194911 0.69 RAB9A (0.51) NPC1RAB9ASMN1; SMN2ALDH1A1HCAR2
SCHEMBL9190029 0.68 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0399856-B1 Pteridin-4 (3H)-ones, processes for their preparation and medicaments containing them LIPHA (FR) 1995-08-09 EP disclosed
US-5270465-A 4(3H)-pteridinone compounds LIPHA, LYONNAISE INDUSTRILLE PHARMACEUTIQUE (FR) 1993-12-14 US disclosed
US-5167949-A Antiallergic LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1992-12-01 US disclosed
EP-0399856-A1 Pteridin-4 (3H)-ones, processes for their preparation and medicaments containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1990-11-28 EP disclosed