SCHEMBL9501020

SCHEMBL9501020

C=CCc1nc2nccnc2c(=O)[nH]1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 5/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
AKR1B1 P15121 1/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
MEN1 O00255 1/20 0.30
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30
ADORA2A P29274 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3817859 0.78 TNKS2 (0.44) HCAR2ALDH1A1HPGDADORA2AL3MBTL1
SCHEMBL9190029 0.74 ALDH1A1 (0.43) HCAR2ALDH1A1
SCHEMBL6440045 0.72 HCAR2 (0.43) HCAR2ALDH1A1HTTL3MBTL1
SCHEMBL9192192 0.71 NPC1 (0.49) HCAR2ALDH1A1KMT2A
SCHEMBL9195013 0.71 HCAR2 (0.37) HCAR2
SCHEMBL9191469 0.71 HCAR2 (0.47) HCAR2ALDH1A1HPGDMEN1KMT2A
SCHEMBL9195100 0.70 RAB9A (0.59) HCAR2MEN1KMT2A
SCHEMBL9194026 0.70 HCAR2 (0.44) HCAR2ALDH1A1
SCHEMBL5332492 0.69 NUDT1 (0.50) NPSR1ALDH1A1HPGD
SCHEMBL9191459 0.69 HCAR2 (0.40) HCAR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5270465-A 4(3H)-pteridinone compounds LIPHA, LYONNAISE INDUSTRILLE PHARMACEUTIQUE (FR) 1993-12-14 US disclosed
US-5167949-A Antiallergic LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1992-12-01 US disclosed
US-3895012-A 2-Alkyl-4(3H)-pteridinone compounds and therapeutic compositions BOEHRINGER MANNHEIM GMBH 1975-07-15 US disclosed
US-3895012-A 2-Alkyl-4(3H)-pteridinone compounds and therapeutic compositions BOEHRINGER MANNHEIM GMBH 1975-07-15 US disclosed