SCHEMBL9192527

SCHEMBL9192527

CC(=O)N(O)C(C)c1cccc(C#Cc2ccc(Cl)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGES O14684 5/20 0.48
AKR1C3 P42330 3/20 0.46
ACACB O00763 1/20 0.41
ASIC3 Q9UHC3 1/20 0.41
ALOX5 P09917 2/20 0.40
EPHX2 P34913 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9192595 0.91 ACACB (0.42) PTGESACACBASIC3ALOX5
SCHEMBL9476083 0.88 ALOX5 (0.52) PTGESAKR1C3ASIC3ALOX5EPHX2
SCHEMBL9189969 0.88 ALOX5 (0.43) PTGESACACBALOX5
SCHEMBL9191848 0.85 PTGES (0.50) PTGESACACBALOX5
SCHEMBL9190507 0.84 PTGES (0.51) PTGESAKR1C3ACACBALOX5EPHX2
SCHEMBL9197190 0.83 PTGES (0.45) PTGESAKR1C3ACACBASIC3ALOX5
SCHEMBL9195594 0.82 ACACB (0.46) PTGESACACBALOX5
SCHEMBL9193333 0.81 PTGES (0.49) PTGESALOX5
SCHEMBL9197314 0.80 ALOX5 (0.36) PTGESALOX5
SCHEMBL4537646 0.79 PTGES (0.50) PTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468281-B1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals GRUENENTHAL GMBH (DE) 1995-03-08 EP disclosed
US-5202349-A Lipoxygenase inhibitors, antiasthatics GRUENENTHAL GMBH (DE) 1993-04-13 US disclosed
EP-0468281-A1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals Grünenthal GmbH (DE) 1992-01-29 EP disclosed