SCHEMBL9192595

SCHEMBL9192595

CC(=O)N(O)C(C)c1cccc(C#Cc2ccc(C(C)C)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.42
FFAR1 O14842 1/20 0.40
PTGES O14684 1/20 0.39
ASIC3 Q9UHC3 1/20 0.39
ALOX5 P09917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9192527 0.91 PTGES (0.48) ACACBPTGESASIC3ALOX5
SCHEMBL9189969 0.89 ALOX5 (0.43) ACACBFFAR1PTGESALOX5
SCHEMBL9195927 0.87 ACACB (0.49) ACACBFFAR1ALOX5
SCHEMBL9191848 0.86 PTGES (0.50) ACACBFFAR1PTGESALOX5
SCHEMBL9190507 0.85 PTGES (0.51) ACACBFFAR1PTGESALOX5
SCHEMBL9195594 0.83 ACACB (0.46) ACACBPTGESALOX5
SCHEMBL9195413 0.83 FFAR1 (0.54) FFAR1ALOX5
SCHEMBL9193333 0.82 PTGES (0.49) FFAR1PTGESALOX5
SCHEMBL9197314 0.81 ALOX5 (0.36) PTGESALOX5
SCHEMBL4537646 0.80 PTGES (0.50) FFAR1PTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468281-B1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals GRUENENTHAL GMBH (DE) 1995-03-08 EP disclosed
US-5202349-A Lipoxygenase inhibitors, antiasthatics GRUENENTHAL GMBH (DE) 1993-04-13 US disclosed
EP-0468281-A1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals Grünenthal GmbH (DE) 1992-01-29 EP disclosed