SCHEMBL9198552

SCHEMBL9198552

Cc1ccc([N+](=O)[O-])c(CN(C(=O)O)[C@H]2C[C@H]3CC[C@@H](C2)N3C)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 5/20 0.42
TP53 P04637 1/20 0.42
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
LMNA P02545 1/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
MAPT P10636 1/20 0.40
GAA P10253 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9198555 1.00 ALDH1A1 (0.42) ALDH1A1KDM4ETP53KMT2AMEN1
SCHEMBL9200033 0.88 NOS3 (0.55) ALDH1A1KDM4EKMT2AMEN1NOS3
SCHEMBL9200027 0.88 NOS3 (0.55) ALDH1A1KDM4EKMT2AMEN1NOS3
SCHEMBL9200471 0.86 KMT2A (0.49) ALDH1A1KDM4EKMT2AMEN1CHRM2
SCHEMBL9200469 0.86 KMT2A (0.49) ALDH1A1KDM4EKMT2AMEN1CHRM2
SCHEMBL9196156 0.86 CHRM1 (0.45) ALDH1A1LMNANOS3NOS1NOS2
SCHEMBL9196158 0.86 CHRM1 (0.45) ALDH1A1LMNANOS3NOS1NOS2
SCHEMBL9203754 0.73 MEN1 (0.41) ALDH1A1KMT2AMEN1CHRM2CHRM1
SCHEMBL9203749 0.73 MEN1 (0.41) ALDH1A1KMT2AMEN1CHRM2CHRM1
SCHEMBL2310221 0.71 MGLL (0.47) ALDH1A1KDM4EKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0382687-B1 Benzofused-N-containing heterocycle derivatives BOEHRINGER INGELHEIM ITALIA (IT) 1995-12-27 EP disclosed
US-5106851-A Respiratory system disorders ISTITUTO DE ANGELI S.P.A. (IT) 1992-04-21 US disclosed
EP-0382687-A2 Benzofused-N-containing heterocycle derivatives BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1990-08-16 EP disclosed