SCHEMBL9199488

SCHEMBL9199488

NCC(CC(=O)O)c1scc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 5/20 0.54
GABBR1 Q9UBS5 5/20 0.54
CYP2C9 P11712 3/20 0.43
LMNA P02545 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
NFKB1 P19838 1/20 0.43
DRD3 P35462 1/20 0.43
BLM P54132 1/20 0.43
CYP2D6 P10635 1/20 0.43
MEN1 O00255 1/20 0.43
THRB P10828 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 1/20 0.43
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
MIF P14174 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL656968 0.78 GABBR2 (0.41) GABBR2GABBR1CYP2C9CYP2C19MEN1
SCHEMBL11040097 0.75 GABBR2 (0.57) GABBR2GABBR1CYP2C9LMNACYP2C19
SCHEMBL9315749 0.73 ALDH1A1 (0.36) CYP2C19CYP1A2BLMMEN1KMT2A
Phenibut SCHEMBL340838 0.71 GABBR2 (1.00) GABBR2GABBR1CYP2C9LMNACYP2C19
Phenibut SCHEMBL351501 0.71 GABBR2 (1.00) GABBR2GABBR1CYP2C9LMNACYP2C19
Phenibut SCHEMBL9545047 0.71 GABBR2 (1.00) GABBR2GABBR1CYP2C9LMNACYP2C19
SCHEMBL2966895 0.71 KMT2A (0.45) CYP2C9CYP1A2MEN1TSHRKMT2A
SCHEMBL354785 0.70 TAAR1 (0.44)
Phenibut SCHEMBL22831453 0.70 GABBR2 (0.96) GABBR2GABBR1CYP2C9LMNACYP2C19
Phenibut SCHEMBL3053795 0.70 GABBR2 (0.96) GABBR2GABBR1CYP2C9LMNACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0463969-B1 New compounds of 4-aminobutyric acid, process for their preparation and pharmaceutical preparations containing them ADIR (FR) 1995-02-08 EP claimed
US-5214063-A 4-aminobutyric acid compounds, compositions and methods of use for treating disorders related to a dysfunction of GABAB receptors ADIR ET COMPAGNIE (FR) 1993-05-25 US disclosed
US-5162364-A Treatment of spastic and senescence disorders ADIR ET COMPAGNIE (FR) 1992-11-10 US disclosed