SCHEMBL9199658

SCHEMBL9199658

CC(=O)N[CH]c1ccc(CBr)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
ALDH1A1 P00352 4/20 0.37
TRPA1 O75762 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 2/20 0.33
TBXAS1 P24557 2/20 0.33
F13A1 P00488 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP2C9 P11712 1/20 0.33
HTT P42858 1/20 0.33
HDAC3 O15379 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
PTPN1 P18031 1/20 0.33
POLB P06746 1/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC2 Q92769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL743446 0.83 HDAC8 (0.45) TSHRKDM4EF13A1KMT2AHDAC3
SCHEMBL295483 0.80 CYP4A11 (0.50) TSHRKDM4EF13A1
SCHEMBL6670487 0.76 ALDH1A1 (0.48) ALDH1A1KDM4EKMT2A
SCHEMBL60234 0.74 AKR1C3 (0.48) ALDH1A1TSHRSMN1; SMN2NPC1RAB9A
SCHEMBL11105167 0.72 AKR1C3 (0.62) CES2CES1ALDH1A1TRPA1TSHR
SCHEMBL11105164 0.72 AKR1C3 (0.62) CES2CES1ALDH1A1TRPA1TSHR
SCHEMBL29638051 0.71 ABCG2 (0.39) CES2CES1ALDH1A1TRPA1SMN1; SMN2
SCHEMBL11641546 0.71 SMN1; SMN2 (0.59) ALDH1A1TSHRSMN1; SMN2NPC1RAB9A
SCHEMBL1501994 0.71 KMT2A (0.63) ALDH1A1SMN1; SMN2NPC1RAB9AKDM4E
SCHEMBL4661731 0.70 TRPA1 (0.39) CES2CES1ALDH1A1TRPA1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0495013-B1 HEXAPEPTIDES WITH SULPHATE ESTER GROUPS FISONS CORP (US) 1995-03-08 EP disclosed
EP-0619823-A1 PEPTIDE COMPOUNDS HAVING THERAPEUTIC ACTIVITY Astra Aktiebolag (SE) 1994-10-19 EP disclosed
EP-0226217-B1 Peptides with sulfate ester group FISONS CORP (US) 1994-01-26 EP disclosed
WO-1993013126-A1 PEPTIDE COMPOUNDS HAVING THERAPEUTIC ACTIVITY FISONS CORPORATION (US) 1993-07-08 WO disclosed