SCHEMBL9199852

SCHEMBL9199852

Cc1cc(-c2cc(Sc3ccc(F)cc3)cc(C(C)C)c2O)ccc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.42
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGS2 P35354 2/20 0.33
BCL2 P10415 2/20 0.33
MCL1 Q07820 2/20 0.33
RPS6KA3 P51812 1/20 0.33
PTGS1 P23219 1/20 0.33
PTPN1 P18031 1/20 0.32
CDC25A P30304 1/20 0.32
CDC25B P30305 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
GCGR P47871 1/20 0.31
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8780227 0.88 HMGCR (0.50) HMGCRMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL9194475 0.82 HMGCR (0.45) HMGCRMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL9193916 0.81 PTGS2 (0.33) PTGS2RPS6KA3PTGS1CA1CA2
SCHEMBL9197287 0.75 HMGCR (0.38) HMGCRMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL9193961 0.73 PTPN5 (0.50) CYP1A2PTGS2RPS6KA3PTGS1CA1
SCHEMBL15177384 0.72 CA1 (0.59) CYP1A2PTGS2RPS6KA3PTGS1CA1
SCHEMBL8780157 0.72 PTGS2 (0.37) HMGCRPTGS2RPS6KA3CA1CA2
SCHEMBL4069702 0.70 HSP90AA1 (0.44) PTGS2RPS6KA3PTGS1AKR1C3AKR1C2
SCHEMBL9512239 0.70 CA1 (0.53) HMGCRCYP1A2RPS6KA3PTGS1CA1
SCHEMBL8780176 0.68 GABRA1 (0.50) HMGCRRPS6KA3CA1CA2GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418648-B1 4-Hydroxytetrahydropyran-2-ones as well as the corresponding dehydroxy carbon acid derivatives, salts and esters, process for their preparation, pharmaceutical preparations as well as precursors HOECHST AG (DE) 1995-01-11 EP disclosed
US-5294724-A Anticholesterol agents HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-15 US disclosed
EP-0418648-A1 4-Hydroxytetrahydropyran-2-ones as well as the corresponding dehydroxy carbon acid derivatives, salts and esters, process for their preparation, pharmaceutical preparations as well as precursors HOECHST AKTIENGESELLSCHAFT (DE) 1991-03-27 EP disclosed