SCHEMBL9201733

SCHEMBL9201733

O=C(O)CC(C[N+](=O)[O-])c1cc2cc(Cl)ccc2o1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.43
KDM4E B2RXH2 3/20 0.43
CYP2C9 P11712 3/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 2/20 0.43
GPR35 Q9HC97 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
POLB P06746 1/20 0.42
MAOB P27338 3/20 0.40
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
ADAM17 P78536 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TSHR P16473 2/20 0.38
MAPT P10636 2/20 0.37
HTT P42858 1/20 0.37
GABBR2 O75899 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9315814 0.84 TP53 (0.48) ALOX5KDM4ECYP2C9ALDH1A1CYP1A2
SCHEMBL9202393 0.82 GABBR2 (0.54) ALOX5KDM4ECYP2C9ALDH1A1CYP1A2
SCHEMBL9201731 0.76 GABBR2 (0.35) CYP2C9ALDH1A1CYP1A2KMT2AMEN1
SCHEMBL27725190 0.74 GABBR2 (0.61) CYP2C9ALDH1A1CYP1A2KMT2AMEN1
SCHEMBL21686411 0.74 GABBR2 (0.61) CYP2C9ALDH1A1CYP1A2KMT2AMEN1
SCHEMBL9988481 0.74 GABBR2 (0.61) CYP2C9ALDH1A1CYP1A2KMT2AMEN1
SCHEMBL657858 0.74 KMT2A (0.48) ALOX5KDM4ECYP2C9ALDH1A1CYP1A2
SCHEMBL9315765 0.71 TAS1R3 (0.41) KDM4EALDH1A1MAOBMMP2MMP9
SCHEMBL9315934 0.70 KDM4E (0.39) KDM4EALDH1A1L3MBTL1MAOBTSHR
SCHEMBL9315905 0.70 CA12 (0.42) KDM4EALDH1A1MAOBTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0463969-B1 New compounds of 4-aminobutyric acid, process for their preparation and pharmaceutical preparations containing them ADIR (FR) 1995-02-08 EP disclosed
EP-0463969-A1 New compounds of 4-aminobutyric acid, process for their preparation and pharmaceutical preparations containing them ADIR ET COMPAGNIE (FR) 1992-01-02 EP disclosed