SCHEMBL9203593

SCHEMBL9203593

CCCc1cccc(C=C(OC(C)C)C(=O)c2ccc(C(=O)N(C)C)cc2)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.34
PDK1 Q15118 4/20 0.33
ALDH1A1 P00352 2/20 0.33
PDK2 Q15119 2/20 0.33
PDK4 Q16654 2/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
PDK3 Q15120 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
LTB4R Q15722 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33
MLYCD O95822 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9200672 0.88 CYP4F2 (0.39) CYP2D6PDK1ALDH1A1PDK2PDK4
SCHEMBL9203046 0.87 CYP4F2 (0.38) CYP2D6PDK1ALDH1A1PDK2PDK4
SCHEMBL9206870 0.86 PTGS2 (0.38) PDK1ALDH1A1PDK2PDK4HPGD
SCHEMBL9206588 0.86 CYP11B1 (0.34) CYP2D6PDK1ALDH1A1PDK2PDK4
SCHEMBL9198641 0.85 NR1H4 (0.36) CYP2D6PDK1ALDH1A1PDK2PDK4
SCHEMBL9202975 0.84 CYP2D6 (0.39) CYP2D6ALDH1A1HPGDSMN1; SMN2ALOX5
SCHEMBL9206423 0.83 HSD17B2 (0.38) CYP2D6ALDH1A1HPGDSMN1; SMN2MAPT
SCHEMBL9204169 0.81 ALDH1A1 (0.41) CYP2D6PDK1ALDH1A1HPGDSMN1; SMN2
SCHEMBL9286479 0.80 ACHE (0.39) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL9208251 0.74 PRSS1 (0.33) ALDH1A1HPGDSMN1; SMN2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed