SCHEMBL9206993

SCHEMBL9206993

Cc1cccc(CCN2CCC(CN3CCc4cc(C)c(C)cc4CC3=O)C2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KDM4E B2RXH2 3/20 0.38
POLB P06746 2/20 0.38
ACHE P22303 2/20 0.37
BCHE P06276 1/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
HTR1A P08908 4/20 0.33
DRD2 P14416 3/20 0.33
HTR2A P28223 2/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPT P10636 1/20 0.33
HCN4 Q9Y3Q4 1/20 0.33
DRD4 P21917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9210290 0.86 KCNH2 (0.41) KCNH2CYP3A4CYP2D6CYP2C19KDM4E
SCHEMBL9206874 0.85 BCHE (0.42) KCNH2CYP3A4KDM4EACHEBCHE
Hydrochloric Acid SCHEMBL9740423 0.85 CYP3A4 (0.42) KCNH2CYP3A4KDM4EACHEBCHE
SCHEMBL9216817 0.81 BCHE (0.38) KCNH2CYP3A4CYP2D6CYP2C19KDM4E
SCHEMBL9204663 0.80 ACHE (0.52) ACHEBCHEMEN1KMT2AHTR1A
SCHEMBL9216033 0.80 ATM (0.39) KDM4EPOLBDRD2ALDH1A1ALOX15
SCHEMBL9207136 0.79 HTR2B (0.39) ACHEBCHEHTR1ADRD2LMNA
SCHEMBL9205651 0.77 HTR1A (0.38) ACHEHTR1ADRD2HTR2ASMN1; SMN2
Hydrochloric Acid SCHEMBL9740530 0.77 CYP3A4 (0.47) KCNH2CYP3A4KDM4EACHEBCHE
SCHEMBL9212638 0.76 ACHE (0.53) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed