SCHEMBL9207261

SCHEMBL9207261

OC(CBr)CCc1cccc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 1/20 0.43
ACP3 P15309 1/20 0.42
SLC18A2 Q05940 1/20 0.41
ADA P00813 1/20 0.41
CYP2D6 P10635 1/20 0.41
CTNNB1 P35222 1/20 0.41
NQO2 P16083 1/20 0.41
DNM1 Q05193 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7277353 0.89 MTNR1A (0.49) MTNR1ATDP1CYP1A2CYP2C19CYP2C9
SCHEMBL8662663 0.87 SIGMAR1 (0.41) MTNR1ATDP1CYP1A2CYP2C19CYP2C9
SCHEMBL8535073 0.84 CYP1A2 (0.50) MTNR1ATDP1CYP1A2CYP2C19CYP2C9
SCHEMBL7278098 0.83 TDP1 (0.47) MTNR1ATDP1CYP1A2CYP2C19CYP2C9
SCHEMBL8539991 0.81 CYP1A2 (0.47) MTNR1ATDP1CYP1A2CYP2C19CYP2C9
SCHEMBL28702695 0.80 SIGMAR1 (0.52) MTNR1ATDP1ACP3CTNNB1
SCHEMBL2480671 0.79 KMT2A (0.51) MTNR1ATDP1CYP1A2CYP2C19CYP2C9
SCHEMBL20825094 0.79 MTNR1A (0.50) MTNR1ATDP1CYP1A2CYP2C19CYP2C9
SCHEMBL6684869 0.78 CYP1A2 (0.48) MTNR1ATDP1CYP1A2CYP2C19CYP2C9
SCHEMBL2692036 0.78 MTNR1A (0.40) MTNR1ATDP1CYP1A2CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed