SCHEMBL9208546

SCHEMBL9208546

COc1cc2c(cc1OC)CC(=O)N(CC1CCN(CCc3csc4ccccc34)C1)CC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 2/20 0.42
MAPT P10636 1/20 0.42
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
HTR1A P08908 3/20 0.39
SLC6A4 P31645 2/20 0.39
CHRM2 P08172 1/20 0.39
DRD3 P35462 1/20 0.39
KCNH2 Q12809 1/20 0.39
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ADRA1B P35368 1/20 0.37
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
ACHE P22303 2/20 0.35
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9208988 0.95 HCN4 (0.41) HCN4MAPTCYP3A4ALOX15HTR1A
SCHEMBL9207815 0.94 HCN4 (0.40) HCN4MAPTCYP3A4ALOX15HTR1A
Hydrochloric Acid SCHEMBL9740138 0.94 CYP3A4 (0.41) HCN4MAPTCYP3A4ALOX15HTR1A
SCHEMBL9205651 0.91 HTR1A (0.38) MAPTHTR1ASLC6A4DRD3SMN1; SMN2
SCHEMBL9214709 0.90 HCN4 (0.41) HCN4MAPTCYP3A4ALOX15HTR1A
SCHEMBL9210593 0.89 HCN4 (0.40) HCN4MAPTCYP3A4ALOX15HTR1A
SCHEMBL9207407 0.88 HTR1A (0.37) HTR1ASLC6A4DRD3SMN1; SMN2DRD4
SCHEMBL9211495 0.86 HTR1A (0.42) MAPTHTR1ASLC6A4SMN1; SMN2BCHE
SCHEMBL9205217 0.86 HCN4 (0.40) HCN4MAPTCYP3A4ALOX15HTR1A
SCHEMBL9213796 0.86 MTNR1A (0.41) HCN4MAPTCYP3A4ALOX15HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed