SCHEMBL9211531

SCHEMBL9211531

COc1ccc(OCCCCl)cc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.57
CA12 O43570 1/20 0.57
CA1 P00915 1/20 0.57
CA7 P43166 1/20 0.57
CA9 Q16790 1/20 0.57
CA14 Q9ULX7 1/20 0.57
MAPT P10636 3/20 0.45
ALDH1A1 P00352 3/20 0.45
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
DRD3 P35462 1/20 0.44
PRSS1 P07477 4/20 0.44
TDP1 Q9NUW8 1/20 0.43
ADRB2 P07550 1/20 0.42
MAPK1 P28482 1/20 0.42
ACHE P22303 2/20 0.42
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7388441 0.93 CA12 (0.53) CA2CA12CA1CA7CA9
SCHEMBL10848385 0.92 CA2 (0.57) CA2CA12CA1CA7CA9
SCHEMBL31570772 0.92 CA2 (0.57) CA2CA12CA1CA7CA9
SCHEMBL1545424 0.87 CA12 (0.61) CA2CA12CA1CA7CA9
SCHEMBL8337382 0.86 CA12 (0.59) CA2CA12CA1CA7CA9
SCHEMBL31648415 0.85 L3MBTL1 (0.46) CA2CA12CA1CA7CA9
SCHEMBL31540368 0.84 ADRB2 (0.49) LMNAADRB2MAPK1ACHETUBB4A
SCHEMBL22498547 0.83 CA2 (0.55) CA2CA12CA1CA7CA9
SCHEMBL16726537 0.83 CA2 (0.55) CA2CA12CA1CA7CA9
SCHEMBL4392307 0.83 CA2 (0.55) CA2CA12CA1CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
US-4950674-A Arylalkylheterocyclic amines,N-substituted by aryloxyalkyl group in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1990-08-21 US disclosed
US-4810713-A Arylalkyl-heterocyclic amines, n-substituted by aryloxyalkyl groups used in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1989-03-07 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed
EP-0235463-A2 N-substituted-arylalkyl and arylalkylene piperidines as cardiovascular antihistaminic and antisecretory agents A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1987-09-09 EP disclosed