SCHEMBL9211545

SCHEMBL9211545

CCOC(=O)c1cc(-c2ccc(S(C)(=O)=O)cc2)n(-c2ccccc2F)n1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.59
CA9 Q16790 3/20 0.58
NR1H2 P55055 1/20 0.52
NPSR1 Q6W5P4 2/20 0.47
TP53 P04637 2/20 0.47
ALDH1A1 P00352 2/20 0.46
PTGS2 P35354 3/20 0.45
PTGS1 P23219 1/20 0.45
FAAH O00519 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9210328 0.89 CHRNA7 (0.63) CHRNA7CA9NR1H2PTGS2PTGS1
SCHEMBL30050028 0.85 NPSR1 (0.51) CHRNA7CA9NPSR1TP53ALDH1A1
SCHEMBL30049915 0.85 NPSR1 (0.51) CHRNA7CA9NPSR1TP53ALDH1A1
SCHEMBL9210036 0.85 CA9 (0.75) CHRNA7CA9NR1H2PTGS2FAAH
SCHEMBL23706283 0.85 NPSR1 (0.51) CHRNA7CA9NPSR1TP53ALDH1A1
SCHEMBL9207359 0.85 ALDH1A1 (0.58) ALDH1A1PTGS2PTGS1
SCHEMBL9208216 0.84 PTGS2 (0.49) CHRNA7NR1H2ALDH1A1PTGS2PTGS1
SCHEMBL7627415 0.83 CHRNA7 (0.83) CHRNA7CA9PTGS2PTGS1
SCHEMBL9941326 0.83 CA9 (0.82) CHRNA7CA9NR1H2PTGS2PTGS1
SCHEMBL7872745 0.83 CHRNA7 (0.66) CHRNA7CA9NR1H2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418845-B1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-09 EP disclosed
EP-0418845-A1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-03-27 EP disclosed