SCHEMBL9211556

SCHEMBL9211556

CC(=O)NCc1ccc(CC2CNCCCNCCCNC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
ACP1 P24666 1/20 0.45
HDAC1 Q13547 2/20 0.43
HDAC6 Q9UBN7 1/20 0.43
ALDH1A1 P00352 3/20 0.42
MAPT P10636 2/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
MC4R P32245 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
JAK3 P52333 1/20 0.38
P2RX7 Q99572 1/20 0.38
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7183846 0.78 GBA1 (0.47) KMT2ASMN1; SMN2
Bromide SCHEMBL7608555 0.75 GBA1 (0.44) KMT2ASMN1; SMN2
SCHEMBL17553578 0.75 CHRNB2 (0.49) KMT2AALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL12133623 0.73 KMT2A (0.76) KMT2AHDAC1HDAC6ALDH1A1MAPT
SCHEMBL10188221 0.72 HTR2C (0.51) KMT2AHDAC1HDAC6ALDH1A1MAPT
Bromide SCHEMBL9096258 0.71 EED (0.41) KMT2AACP1
SCHEMBL9015445 0.71 GBA1 (0.41) KMT2AALDH1A1MAPT
SCHEMBL30589132 0.71 GBA1 (0.61) KMT2APOLB
SCHEMBL15918525 0.70 ALDH1A1 (0.51) KMT2AHDAC1HDAC6ALDH1A1SMN1; SMN2
SCHEMBL20808158 0.70 L3MBTL1 (0.46) HDAC1ALDH1A1MAPTSMN1; SMN2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0329737-B1 TRI-AZA MACROCYCLES AND METAL COMPLEXES THEREOF CELLTECH THERAPEUTICS LTD (GB) 1995-04-12 EP disclosed
US-5247075-A Imaging agents, cytotoxic agents CELLTECH LIMITED (GB) 1993-09-21 US disclosed
EP-0329737-A1 TRI-AZA MACROCYCLES AND METAL COMPLEXES THEREOF CELLTECH THERAPEUTICS LIMITED (GB) 1989-08-30 EP disclosed
WO-1989001475-A1 TRI-AZA MACROCYCLES AND METAL COMPLEXES THEREOF CELLTECH LIMITED (GB) 1989-02-23 WO disclosed