SCHEMBL9211774

SCHEMBL9211774

Cc1ccc(S(=O)(=O)OCC2=C3C=CC=CC3C=Cc3ccccc32)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VDR P11473 2/20 0.37
DHODH Q02127 1/20 0.35
ALDH1A1 P00352 4/20 0.34
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 2/20 0.31
HPGD P15428 1/20 0.31
MAPT P10636 2/20 0.31
USP2 O75604 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
NOD2 Q9HC29 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
STAT3 P40763 1/20 0.30
F2 P00734 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9205978 0.83 VDR (0.34) VDRDHODHALDH1A1KEAP1NFE2L2
SCHEMBL13954243 0.68 VDR (0.51) VDRDHODHALDH1A1KEAP1NFE2L2
SCHEMBL9684266 0.68 VDR (0.48) VDRDHODHALDH1A1KEAP1NFE2L2
SCHEMBL8061919 0.66 VDR (0.47) VDRALDH1A1KEAP1NFE2L2MEN1
SCHEMBL29995677 0.65 SYK (0.50) ALDH1A1KMT2AKDM4EMAPTLMNA
SCHEMBL3777059 0.65 SYK (0.50) ALDH1A1KMT2AKDM4EMAPTLMNA
SCHEMBL2890 0.65 CA9 (0.53) VDRALDH1A1KMT2AMAPTLMNA
Toluene SCHEMBL9257721 0.64 CA9 (0.51) VDRALDH1A1MAPTLMNACYP2C9
Ammonia Solution, Strong SCHEMBL9470841 0.64 CA9 (0.51) VDRALDH1A1KMT2AMAPTLMNA
SCHEMBL8734172 0.63 HTR6 (0.37) VDRALDH1A1KEAP1NFE2L2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0319073-B1 Cyclo-octane neuroprotective agents MERCK SHARP & DOHME (GB) 1995-08-23 EP disclosed
US-4927819-A ANTICONVULSANT, PREVENTION OF NEURODEGENERATIVE DISORDERS MERCK SHARP & DOHME LIMITED (GB) 1990-05-22 US disclosed
EP-0319073-A2 Cyclo-octane neuroprotective agents MERCK SHARP & DOHME LTD. (GB) 1989-06-07 EP disclosed