SCHEMBL9212660

SCHEMBL9212660

C=CCN1C[C@H](C)N(c2c(O)cccc2Cc2cccc(C(=O)N(CC)c3ccccc3)c2)C[C@H]1C

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
HPGD P15428 2/20 0.41
CYP2C19 P33261 2/20 0.41
OPRD1 P41143 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6915923 0.86 OPRD1 (0.43) CYP1A2CYP3A4CYP2C9HPGDOPRD1
SCHEMBL4576511 0.84 OPRD1 (0.59) OPRD1
SCHEMBL8930490 0.84 OPRD1 (0.40) CYP1A2CYP3A4OPRD1
SCHEMBL7993545 0.81 CYP3A4 (0.54) KDM4ECYP1A2CYP3A4CYP2C9HPGD
SCHEMBL4591245 0.81 CYP3A4 (0.54) KDM4ECYP1A2CYP3A4CYP2C9HPGD
SCHEMBL8009424 0.81 CYP3A4 (0.54) KDM4ECYP1A2CYP3A4CYP2C9HPGD
SCHEMBL8002856 0.81 CYP3A4 (0.54) KDM4ECYP1A2CYP3A4CYP2C9HPGD
SCHEMBL5146343 0.76 OPRD1 (0.45) HPGDOPRD1
SCHEMBL8930486 0.75 OPRD1 (0.55) OPRD1
SCHEMBL8930450 0.73 OPRD1 (0.72) CYP1A2CYP3A4CYP2C9HPGDOPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995004051-A1 PIPERAZINE COMPOUNDS USED IN THERAPY THE WELLCOME FOUNDATION LIMITED (GB) 1995-02-09 WO disclosed