SCHEMBL9212860

SCHEMBL9212860

ClCC1CCCCN(CCCOc2ccc3c(c2)OCO3)C1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.57
KCNH2 Q12809 2/20 0.57
MEN1 O00255 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
MAPT P10636 1/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.53
MAPK1 P28482 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
RAB9A P51151 2/20 0.47
POLB P06746 1/20 0.47
MAOB P27338 4/20 0.46
MAOA P21397 1/20 0.44
FAAH O00519 2/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9741229 0.80 RAB9A (0.51) MEN1MAPK1KMT2ATDP1RAB9A
SCHEMBL9217121 0.79 HRH3 (0.56) HRH3KCNH2MAPTPOLB
SCHEMBL9278988 0.79 HRH3 (0.48) HRH3KCNH2
SCHEMBL9217118 0.79 DRD2 (0.49) HRH3KCNH2MEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9738996 0.78 HRH3 (0.48) HRH3KCNH2MEN1CYP1A2CYP3A4
SCHEMBL9206438 0.78 HRH3 (0.64) HRH3TSHRKMT2A
SCHEMBL9215679 0.78 KDM4E (0.67) HRH3TSHRKMT2A
SCHEMBL7398551 0.78 HRH3 (0.73) HRH3KCNH2MEN1CYP1A2CYP3A4
SCHEMBL9699038 0.77 MAOB (0.49) HRH3KCNH2MEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9528708 0.77 RAB9A (0.50) HRH3KCNH2MEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed