SCHEMBL9214818

SCHEMBL9214818

Cc1cc2c(cc1C)C(=O)N(CC1CCN(CCc3ccc4ccccc4c3)C1)CC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.42
HTR1A P08908 1/20 0.42
HRH3 Q9Y5N1 3/20 0.41
GRM5 P41594 2/20 0.40
ACHE P22303 2/20 0.39
SIGMAR1 Q99720 3/20 0.37
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
KCNJ1 P48048 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739700 0.95 GRM5 (0.41) SLC6A4HTR1AHRH3GRM5ACHE
SCHEMBL9213420 0.93 HRH3 (0.46) SLC6A4HTR1AHRH3GRM5SIGMAR1
SCHEMBL9207074 0.89 GRM5 (0.42) HRH3GRM5SIGMAR1
Hydrochloric Acid SCHEMBL9213427 0.89 GRM5 (0.42) HRH3GRM5SIGMAR1
SCHEMBL9215099 0.88 ADRA1B (0.46) SLC6A4HTR1AHRH3ACHESIGMAR1
SCHEMBL9215558 0.88 GRM5 (0.41) HRH3GRM5SIGMAR1HDAC3HDAC4
Hydrochloric Acid SCHEMBL9209695 0.88 ADRA1B (0.46) SLC6A4HTR1AACHE
SCHEMBL9215483 0.84 HTR1A (0.44) SLC6A4HTR1A
Bromide SCHEMBL9206535 0.84 KDM2B (0.39) SLC6A4HTR1AACHE
Hydrochloric Acid SCHEMBL9213668 0.83 ABCB1 (0.46) SLC6A4HTR1AGRM5ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed