SCHEMBL9215558

SCHEMBL9215558

Cc1cc2c(cc1C)C(=O)N(CC1CCCCCN(CCCc3ccc4ccccc4c3)C1)CC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.41
HRH3 Q9Y5N1 4/20 0.40
SIGMAR1 Q99720 4/20 0.39
BCHE P06276 1/20 0.38
CHRNB2 P17787 2/20 0.35
CHRNB4 P30926 2/20 0.35
CHRNA3 P32297 2/20 0.35
CHRNA4 P43681 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
PRMT5 O14744 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9207074 0.97 GRM5 (0.42) GRM5HRH3SIGMAR1CHRNB2CHRNB4
Hydrochloric Acid SCHEMBL9213427 0.96 GRM5 (0.42) GRM5HRH3SIGMAR1CHRNB2CHRNB4
SCHEMBL9213420 0.95 HRH3 (0.46) GRM5HRH3SIGMAR1BCHEPRMT5
SCHEMBL9739700 0.93 GRM5 (0.41) GRM5HRH3SIGMAR1HDAC3HDAC4
SCHEMBL9213761 0.90 CHRNB2 (0.43) GRM5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9214818 0.88 SLC6A4 (0.42) GRM5HRH3SIGMAR1HDAC3HDAC4
SCHEMBL9740802 0.86 SIGMAR1 (0.45) GRM5SIGMAR1BCHECHRNB2CHRNB4
Hydrochloric Acid SCHEMBL9208899 0.85 CHRNB2 (0.46) GRM5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9215804 0.83 GRM5 (0.39) GRM5HRH3CHRNB2CHRNB4CHRNA3
SCHEMBL9208130 0.82 HRH3 (0.44) GRM5HRH3SIGMAR1PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed