SCHEMBL9215673

SCHEMBL9215673

COc1cc2c(cc1OC)CC(=O)N(CC1CCN(CCCc3c[nH]c4ccccc34)C1)C=C2

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.45
PDE4D Q08499 5/20 0.44
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
HTR1D P28221 2/20 0.42
HTR1B P28222 2/20 0.42
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9742174 0.87 HTR1A (0.43) HTR1AHTR1DHTR1BDRD2
SCHEMBL9216571 0.84 PDE4D (0.49) HTR1APDE4DPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL9740012 0.82 PDE4D (0.48) HTR1APDE4DPDE4APDE4BPDE4C
Hydrochloric Acid SCHEMBL9207604 0.81 HTR1A (0.52) HTR1APDE4DHTR1DHTR1BDRD2
SCHEMBL9215863 0.79 BRD4 (0.40) PDE4D
Hydrochloric Acid SCHEMBL9741187 0.79 PDE4D (0.48) HTR1APDE4DPDE4APDE4BPDE4C
SCHEMBL9215979 0.79 PDE4D (0.48) HTR1APDE4DPDE4APDE4BPDE4C
SCHEMBL10894643 0.79 HCN4 (0.48) PDE4DPDE4APDE4BPDE4C
Water SCHEMBL9740391 0.78 PDE4D (0.47) HTR1APDE4DPDE4APDE4BPDE4C
SCHEMBL9739670 0.78 HCN4 (0.55) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed