SCHEMBL9216358

SCHEMBL9216358

COc1cc2c(cc1OC)C(=O)N(CC1CCCN(Cc3ccncc3)C1)CC2

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.49
ADRA1B P35368 1/20 0.44
PDE4D Q08499 3/20 0.43
ACHE P22303 4/20 0.43
HTR1A P08908 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GRM5 P41594 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9215814 0.98 PDE4B (0.48) PDE4BADRA1BPDE4DACHEHTR1A
SCHEMBL9208530 0.91 BCHE (0.50) PDE4DACHEDRD4GRM5MAOB
Hydrochloric Acid SCHEMBL9211501 0.88 ALDH1A1 (0.49) ADRA1BACHEMEN1KMT2AMAOA
SCHEMBL9207082 0.87 BCHE (0.48) PDE4DACHEDRD4GRM5MAOB
SCHEMBL9215461 0.85 BCHE (0.56) PDE4DACHEDRD4MAOB
SCHEMBL9739479 0.82 ADRA1B (0.46) ADRA1BACHEHTR1ADRD4DRD3
SCHEMBL9208347 0.81 ADRA1B (0.48) ADRA1BMEN1KMT2A
Hydrochloric Acid SCHEMBL10644273 0.81 PDE4B (0.66) PDE4BKMT2A
Hydrochloric Acid SCHEMBL9214600 0.81 ADRA1B (0.47) ADRA1BMEN1KMT2A
Hydrochloric Acid SCHEMBL9214568 0.80 PDE4B (0.64) PDE4BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed