SCHEMBL9208530

SCHEMBL9208530

COc1cc2c(cc1OC)C(=O)N(CC1CCCN(Cc3ccccc3)C1)CC2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.50
ACHE P22303 3/20 0.50
FAAH O00519 1/20 0.50
ABCC4 O15439 1/20 0.50
CACNA1F O60840 1/20 0.50
PDE5A O76074 1/20 0.50
ABCB11 O95342 1/20 0.50
APP P05067 1/20 0.50
CHRM2 P08172 1/20 0.50
ABCB1 P08183 1/20 0.50
CYP3A4 P08684 1/20 0.50
CHRM5 P08912 1/20 0.50
ADRA2A P08913 1/20 0.50
CHRM1 P11229 1/20 0.50
ADRA2C P18825 1/20 0.50
DRD4 P21917 1/20 0.50
SLC6A2 P23975 1/20 0.50
MAOB P27338 1/20 0.50
AGTR1 P30556 1/20 0.50
ADRA1A P35348 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9207082 0.96 BCHE (0.48) BCHEACHEFAAHABCC4CACNA1F
SCHEMBL9215461 0.94 BCHE (0.56) BCHEACHEFAAHABCC4CACNA1F
SCHEMBL9216358 0.91 PDE4B (0.49) ACHEDRD4MAOBPDE4DGRM5
Hydrochloric Acid SCHEMBL9211501 0.90 ALDH1A1 (0.49) ACHEMAOBKDM4E
Hydrochloric Acid SCHEMBL9215814 0.89 PDE4B (0.48) BCHEACHEDRD4PDE4DKDM4E
SCHEMBL9739479 0.83 ADRA1B (0.46) ACHEABCB1DRD4GRM5
SCHEMBL9207113 0.83 HTT (0.52) BCHEACHEFAAHABCC4CACNA1F
SCHEMBL9208347 0.83 ADRA1B (0.48) CYP3A4SIGMAR1KDM4E
Hydrochloric Acid SCHEMBL9213957 0.83 HTT (0.51) BCHEACHEDRD4KDM4EGRM5
SCHEMBL9739815 0.82 FAAH (0.45) BCHEACHEFAAHABCC4CACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed