SCHEMBL9216967

SCHEMBL9216967

COc1ccc2cc(CCN3CCCCC3CCN3CCc4cc(C)c(C)cc4C3=O)ccc2c1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 11/20 0.37
TRPV6 Q9H1D0 1/20 0.37
DRD2 P14416 2/20 0.37
DRD4 P21917 1/20 0.37
SIGMAR1 Q99720 2/20 0.36
GPR84 Q9NQS5 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9206975 0.88 ALDH1A1 (0.35) HRH3TRPV6DRD2DRD4
SCHEMBL9208020 0.83 HCN4 (0.49) HRH3TRPV6
Hydrochloric Acid SCHEMBL9739344 0.82 CYP3A4 (0.49) HRH3TRPV6
Hydrochloric Acid SCHEMBL9207084 0.81 ADRA1B (0.39) DRD4
Hydrochloric Acid SCHEMBL9206844 0.81 CYP3A4 (0.47) DRD4
Hydrochloric Acid SCHEMBL9212120 0.78 DRD4 (0.42) HRH3DRD2DRD4
Hydrochloric Acid SCHEMBL9739509 0.76 CYP3A4 (0.49) HRH3
Hydrochloric Acid SCHEMBL9739342 0.73 CYP3A4 (0.49)
SCHEMBL11737839 0.73 SIGMAR1 (0.48) HRH3TRPV6SIGMAR1
SCHEMBL9217265 0.72 DRD4 (0.43) HRH3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed