SCHEMBL9217149

SCHEMBL9217149

CO/C(=N\C#N)c1ccc(C#N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.41
CA1 P00915 2/20 0.41
ALDH1A1 P00352 3/20 0.40
MAPT P10636 1/20 0.40
POLB P06746 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
LMNA P02545 2/20 0.39
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
CYP2A6 P11509 1/20 0.39
CA12 O43570 1/20 0.39
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
PARP15 Q460N3 1/20 0.39
PARP10 Q53GL7 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
GSK3B P49841 2/20 0.38
LOXL2 Q9Y4K0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9217151 1.00 CA2 (0.41) CA2CA1ALDH1A1MAPTPOLB
SCHEMBL30827437 0.81 GSK3B (0.40) ALDH1A1MAPTRXFP1LMNAGSK3B
SCHEMBL9532199 0.81 RAB9A (0.38) ALDH1A1MAPTLMNAHTTKDM4E
SCHEMBL3455077 0.81 POLB (0.52) ALDH1A1MAPTPOLBLMNAHTT
SCHEMBL3455076 0.81 POLB (0.52) ALDH1A1MAPTPOLBLMNAHTT
SCHEMBL9532178 0.78 SMN1; SMN2 (0.37) ALDH1A1MAPTLMNACYP2A6KDM4E
SCHEMBL9532175 0.78 SMN1; SMN2 (0.37) ALDH1A1MAPTLMNACYP2A6KDM4E
SCHEMBL9211615 0.71 MAPT (0.40) ALDH1A1MAPTPOLBLMNAHTT
SCHEMBL9211646 0.71 CYP3A4 (0.35) ALDH1A1MAPTPOLBKDM4EMEN1
SCHEMBL9211650 0.71 CYP3A4 (0.35) ALDH1A1MAPTPOLBKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP disclosed
US-5272164-A Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1993-12-21 US disclosed
US-5223508-A Hypotensive agents, vasodilators KIRIN BEER KABUSHIKI KAISHA (JP) 1993-06-29 US disclosed
US-5166347-A Hypotensive agents, cardiovascular disorders, antiischemic agents and anticoagulants KIRIN BEER KABUSHIKI KAISHA (JP) 1992-11-24 US disclosed
EP-0388528-A2 Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1990-09-26 EP disclosed