SCHEMBL9217306

SCHEMBL9217306

COc1cc2c(cc1OC)C(=O)N(CC1CCCCN(CCc3cccc4ccccc34)C1)CC2

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA1B P35368 1/20 0.46
HTR1A P08908 2/20 0.42
SLC6A4 P31645 1/20 0.42
GRM5 P41594 1/20 0.41
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ABCB1 P08183 1/20 0.39
ABCC1 P33527 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9209429 0.99 ADRA1B (0.45) ADRA1BHTR1ASLC6A4GRM5DRD4
Hydrochloric Acid SCHEMBL9214810 0.97 ADRA1B (0.46) ADRA1BHTR1ASLC6A4GRM5MEN1
Hydrochloric Acid SCHEMBL9213070 0.89 ADRA1B (0.41) ADRA1BGRM5HCRTR1HCRTR2ABCB1
Hydrochloric Acid SCHEMBL9213413 0.88 ADRA1B (0.41) ADRA1BGRM5HCRTR1HCRTR2MEN1
SCHEMBL9208286 0.87 ADRA1B (0.41) ADRA1BGRM5HCRTR1HCRTR2ABCB1
Hydrochloric Acid SCHEMBL9214235 0.87 ADRA1B (0.41) ADRA1BGRM5HCRTR1HCRTR2ABCB1
Hydrochloric Acid SCHEMBL9209655 0.85 GRM5 (0.39) ADRA1BHTR1ASLC6A4GRM5HRH3
Hydrochloric Acid SCHEMBL9207178 0.85 ADRA1B (0.41) ADRA1BGRM5HCRTR1HCRTR2MEN1
SCHEMBL9740802 0.84 SIGMAR1 (0.45) GRM5
SCHEMBL9212922 0.83 HTT (0.49) ADRA1BHTR1AGRM5DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed