Sucrosofate

Sucrosofate

SCHEMBL921799

N.N.N.N.N.N.N.N.O=S(=O)(O)OC[C@H]1O[C@@](COS(=O)(=O)O)(O[C@H]2O[C@H](COS(=O)(=O)O)[C@@H](OS(=O)(=O)O)[C@H](OS(=O)(=O)O)[C@H]2OS(=O)(=O)O)[C@@H](OS(=O)(=O)O)[C@@H]1OS(=O)(=O)O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

TOP1

The experimentally established mechanism targets of Sucrosofate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FGF1 P05230 6/20 0.72
FGF2 P09038 4/20 0.72
SERPINC1 P01008 1/20 0.36
HPSE Q9Y251 13/20 0.35
VEGFA P15692 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sucrosofate SCHEMBL145069 0.99 FGF1 (0.74) FGF1FGF2SERPINC1HPSEVEGFA
Sucrosofate SCHEMBL145070 0.99 FGF1 (0.74) FGF1FGF2SERPINC1HPSEVEGFA
Sucrosofate SCHEMBL16661862 0.99 FGF1 (0.74) FGF1FGF2SERPINC1HPSEVEGFA
Sucrosofate SCHEMBL18467935 0.99 FGF1 (0.74) FGF1FGF2SERPINC1HPSEVEGFA
Sucrosofate SCHEMBL16661861 0.99 FGF1 (0.74) FGF1FGF2SERPINC1HPSEVEGFA
Sucrosofate SCHEMBL18742107 0.98 FGF1 (0.72) FGF1FGF2SERPINC1HPSEVEGFA
Sucrosofate SCHEMBL18244210 0.92 FGF1 (0.65) FGF1FGF2SERPINC1HPSEVEGFA
Sucrosofate SCHEMBL19358882 0.92 FGF1 (0.65) FGF1FGF2SERPINC1HPSEVEGFA
Sucrosofate SCHEMBL2063889 0.92 FGF1 (0.65) FGF1FGF2SERPINC1HPSEVEGFA
Water SCHEMBL41379 0.89 FGF1 (0.61) FGF1FGF2SERPINC1HPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117750944-A Vinorelbine tartrate liposome and raw material composition, preparation method and application thereof 上海济煜医药科技有限公司 2024-03-22 CN claimed
WO-2023051799-A1 VINORELBINE TARTRATE LIPOSOME, AND RAW MATERIAL COMPOSITION THEREOF, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF 上海济煜医药科技有限公司 2023-04-06 WO claimed
CN-103181897-B Gefitinib liposome preparation and preparation method thereof UNIV SHENYANG PHARMACEUTICAL 2015-06-10 CN claimed
CN-102485212-B Sunitinib malate liposome and preparation method thereof UNIV SHENYANG PHARMACEUTICAL 2014-04-09 CN claimed
CN-103181897-A Gefitinib liposome preparation and preparation method thereof UNIV SHENYANG PHARMACEUTICAL 2013-07-03 CN claimed
CN-102805729-A Vinflunine liposome preparation and preparation method of vinflunine liposome preparation QILU PHARMACEUTICAL CO LTD 2012-12-05 CN claimed
CN-102485212-A Sunitinib malate liposome and preparation method thereof UNIV SHENYANG PHARMACEUTICAL 2012-06-06 CN claimed
US-4990610-A Reacting Sucrose with Chlorosulfonic acid and 2-Picoline APPLIED ANALYTICAL INDUSTRIES, INC. (US) 1991-02-05 US claimed
WO-1990002133-A1 METHOD FOR PREPARING SUCRALFATE AND AAI-10001 FORMULATIONS DEVELOPMENT LABORATORIES, INC. (US) 1990-03-08 WO claimed
CN-117750944-A Vinorelbine tartrate liposome and raw material composition, preparation method and application thereof 上海济煜医药科技有限公司 2024-03-22 CN disclosed
WO-2023190709-A1 LIPOSOME COMPOSITION AND LIPOSOME-CONTAINING PHARMACEUTICAL COMPOSITION エーザイ・アール・アンド・ディー・マネジメント株式会社 2023-10-05 WO disclosed
US-11771651-B2 Liposomes and uses thereof ACADEMIA SINICA (TW) 2023-10-03 US disclosed
WO-2023072890-A1 PROCESS FOR THE PREPARATION OF SUCROSE OCTASULFATE OCTAKISTRIETHYLAMMONIUM SALT (TASOS) POWDER AND USES THEREOF SANDOZ AG (CH) 2023-05-04 WO disclosed
EP-4169928-A1 PROCESS FOR THE PREPARATION OF SUCROSE OCTASULFATE OCTAKISTRIETHYLAMMONIUM SALT (TASOS) POWDER AND USES THEREOF SANDOZ AG (CH) 2023-04-26 EP disclosed
EP-0691976-A1 ANTICOAGULANT COMPOUNDS QUEEN'S UNIVERSITY AT KINGSTON (CA) 1996-01-17 EP disclosed
WO-1994022885-A1 ANTICOAGULANT COMPOUNDS QUEEN'S UNIVERSITY AT KINGSTON (CA) 1994-10-13 WO disclosed
WO-1994022437-A2 METHOD FOR TREATING AMYLOIDOSIS QUEEN'S UNIVERSITY AT KINGSTON (CA) 1994-10-13 WO disclosed
US-5084446-A Reaction of aluminum chlorohydrate and sucrose octaammonium sulfate APPLIED ANALYTICAL INDUSTRIES, INC. (US) 1992-01-28 US disclosed
US-4990610-A Reacting Sucrose with Chlorosulfonic acid and 2-Picoline APPLIED ANALYTICAL INDUSTRIES, INC. (US) 1991-02-05 US disclosed
WO-1990002133-A1 METHOD FOR PREPARING SUCRALFATE AND AAI-10001 FORMULATIONS DEVELOPMENT LABORATORIES, INC. (US) 1990-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11771651-B2 Liposomes and uses thereof LYPLAL1, SMPD1, LGMN FGF1 4326/4885FGF2 4197/4885SERPINC1 3060/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.