SCHEMBL9218291

SCHEMBL9218291

BrCc1nc(-c2cc3ccccc3cn2)cc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
CYP1A2 P05177 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ADORA3 P0DMS8 1/20 0.42
RAB9A P51151 1/20 0.41
GRM4 Q14833 5/20 0.39
TDP1 Q9NUW8 1/20 0.39
BTK Q06187 1/20 0.39
CYP2A6 P11509 1/20 0.38
PDPK1 O15530 1/20 0.38
MIF P14174 1/20 0.37
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GPR3 P46089 1/20 0.34
NPY5R Q15761 1/20 0.33
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9494876 0.88 ADORA3 (0.45) NPC1CYP1A2ADORA3RAB9ATDP1
SCHEMBL10510673 0.78 ADORA3 (0.44) CYP1A2KDM4EADORA3IDO1TDO2
SCHEMBL5470573 0.76 NPC1 (0.63) NPC1CYP1A2KDM4ERAB9AGRM4
SCHEMBL31427619 0.72 ALDH1A1 (0.37) CYP1A2KDM4EADORA3TDP1CYP2A6
SCHEMBL28328752 0.70 L3MBTL1 (0.44) CYP1A2KDM4ECYP2A6L3MBTL1
Bromide SCHEMBL5045247 0.69 ALDH1A1 (0.34) CYP1A2ADORA3TDP1CYP2A6L3MBTL1
SCHEMBL31427616 0.68 ALDH1A1 (0.33) CYP1A2ADORA3L3MBTL1
SCHEMBL29526856 0.67 ATM (0.51) NPC1CYP1A2KDM4ERAB9ATDP1
SCHEMBL1169875 0.67 ATM (0.51) NPC1CYP1A2KDM4ERAB9ATDP1
SCHEMBL731645 0.67 NPC1 (0.62) NPC1CYP1A2KDM4ERAB9AGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0180492-A1 Macropolycyclic complexes of rare earth metals and application as fluorescent labels CIS BIO INTERNATIONAL (FR) 1986-05-07 EP claimed
US-5432101-A Complex consists of biologically active molecule associated by coupling or adsorption with the complex COMPAGNIE ORIS INDUSTRIE SA (FR) 1995-07-11 US disclosed
US-5220012-A Macropolycyclic rare earth complexes and application as fluorescent tracers COMPAGNIE ORIS INDUSTRIE SA (FR) 1993-06-15 US disclosed
US-4927923-A IMMUNOLOGY COMPAGNIE ORIS INDUSTRIES (FR) 1990-05-22 US disclosed