SCHEMBL9218686

SCHEMBL9218686

N#CN=C(Nc1ccccc1)c1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.51
TAAR1 Q96RJ0 1/20 0.46
KMT2A Q03164 2/20 0.44
JAK2 O60674 1/20 0.44
TYK2 P29597 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 2/20 0.43
CA9 Q16790 2/20 0.43
CA1 P00915 1/20 0.43
KCNK3 O14649 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.40
BCHE P06276 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
POLB P06746 2/20 0.40
STAT3 P40763 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9215336 0.76 NPC1 (0.53) HTTKMT2AALDH1A1KCNK3SMN1; SMN2
SCHEMBL9213657 0.73 RAB9A (0.48) KMT2AALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL9213141 0.72 RAB9A (0.50) HTTKMT2AALDH1A1SMN1; SMN2CYP3A4
SCHEMBL14257373 0.71 LMNA (0.44) HTTTAAR1KMT2AJAK2TYK2
SCHEMBL9273043 0.71 LMNA (0.44) HTTTAAR1KMT2AJAK2TYK2
SCHEMBL11156357 0.70 RAB9A (0.57) KMT2AALDH1A1GAACYP1A2CYP3A4
SCHEMBL160935 0.69 MDM2 (0.44) TAAR1KMT2AJAK2TYK2ALDH1A1
SCHEMBL15366862 0.69 MDM2 (0.44) TAAR1KMT2AJAK2TYK2ALDH1A1
SCHEMBL6947269 0.69 MDM2 (0.44) TAAR1KMT2AJAK2TYK2ALDH1A1
SCHEMBL11157132 0.69 ROCK1 (0.52) HTTALDH1A1GAACA9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP claimed
US-5223508-A Hypotensive agents, vasodilators KIRIN BEER KABUSHIKI KAISHA (JP) 1993-06-29 US claimed
EP-0388528-A2 Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1990-09-26 EP claimed
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP disclosed
US-5272164-A Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1993-12-21 US disclosed
US-5223508-A Hypotensive agents, vasodilators KIRIN BEER KABUSHIKI KAISHA (JP) 1993-06-29 US disclosed
US-5166347-A Hypotensive agents, cardiovascular disorders, antiischemic agents and anticoagulants KIRIN BEER KABUSHIKI KAISHA (JP) 1992-11-24 US disclosed
EP-0388528-A2 Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1990-09-26 EP disclosed