SCHEMBL9213141

SCHEMBL9213141

Cc1ccc(NC(=NC#N)c2cccnc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.50
NPC1 O15118 3/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C19 P33261 2/20 0.50
NAMPT P43490 2/20 0.50
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
KMT2A Q03164 4/20 0.46
TDP1 Q9NUW8 2/20 0.45
MAPT P10636 2/20 0.44
GFER P55789 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PSMD14 O00487 1/20 0.44
POLB P06746 1/20 0.44
HTT P42858 1/20 0.43
TP53 P04637 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9218840 0.83 NAMPT (0.49) RAB9ANAMPTALDH1A1SMN1; SMN2KMT2A
SCHEMBL1971026 0.75 NAMPT (0.78) RAB9ANPC1CYP3A4NAMPTALDH1A1
SCHEMBL9502986 0.74 THRB (0.45) RAB9ANPC1CYP3A4CYP2C19ALDH1A1
SCHEMBL9213133 0.74 KMT2A (0.42) RAB9ANPC1CYP3A4CYP2C19NAMPT
SCHEMBL9218629 0.74 KMT2A (0.42) RAB9ANPC1CYP3A4CYP2C19NAMPT
SCHEMBL9216085 0.73 RAB9A (0.41) RAB9ANPC1CYP3A4CYP2C19ALDH1A1
SCHEMBL9211594 0.72 KEAP1 (0.52) RAB9ANPC1CYP3A4CYP2C19NAMPT
SCHEMBL9212192 0.72 CFTR (0.44) CYP2C19ALDH1A1SMN1; SMN2KMT2APOLB
SCHEMBL9218686 0.72 HTT (0.51) CYP3A4CYP2C19NAMPTALDH1A1SMN1; SMN2
SCHEMBL9528709 0.72 ALDH1A1 (0.51) CYP3A4CYP2C19ALDH1A1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP claimed
US-5223508-A Hypotensive agents, vasodilators KIRIN BEER KABUSHIKI KAISHA (JP) 1993-06-29 US claimed
EP-0388528-A2 Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1990-09-26 EP claimed
EP-0388528-B1 Carboximidamide derivatives KIRIN BREWERY (JP) 1995-09-27 EP disclosed
US-5272164-A Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1993-12-21 US disclosed
US-5223508-A Hypotensive agents, vasodilators KIRIN BEER KABUSHIKI KAISHA (JP) 1993-06-29 US disclosed
US-5166347-A Hypotensive agents, cardiovascular disorders, antiischemic agents and anticoagulants KIRIN BEER KABUSHIKI KAISHA (JP) 1992-11-24 US disclosed
EP-0388528-A2 Carboximidamide derivatives KIRIN BEER KABUSHIKI KAISHA (JP) 1990-09-26 EP disclosed