SCHEMBL9218755

SCHEMBL9218755

COc1ccc(-c2ccncc2)cc1C#N

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
USP2 O75604 1/20 0.53
F11 P03951 1/20 0.47
CYP17A1 P05093 1/20 0.47
PIK3CD O00329 1/20 0.46
PIK3CA P42336 1/20 0.46
PIK3CB P42338 1/20 0.46
CYP3A4 P08684 1/20 0.46
AAK1 Q2M2I8 1/20 0.46
PRKACA P17612 1/20 0.46
CDK8 P49336 1/20 0.46
CLK2 P49760 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
CDK9 P50750 1/20 0.46
CDK5 Q00535 1/20 0.46
PRKCQ Q04759 1/20 0.46
ROCK1 Q13464 1/20 0.46
DYRK1A Q13627 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025473 0.89 CTSD (0.52) ALDH1A1KDM4ECYP17A1CYP11B1CYP11B2
SCHEMBL29123961 0.83 MAOB (0.57) ALDH1A1KDM4EUSP2F11IMPDH2
SCHEMBL9215557 0.81 CTSD (0.55) ALDH1A1KDM4EUSP2CYP17A1CYP11B1
SCHEMBL5326742 0.81 ALDH1A1 (0.54) ALDH1A1KDM4EUSP2F11IMPDH2
SCHEMBL16158576 0.79 ALDH1A1 (0.51) ALDH1A1KDM4EUSP2F11GSK3B
SCHEMBL11330797 0.78 MAPT (0.61) ALDH1A1CYP17A1PIK3CA
SCHEMBL25543963 0.77 PIK3CD (0.46) ALDH1A1KDM4EPIK3CDPIK3CAPIK3CB
SCHEMBL25544693 0.77 PIK3CD (0.46) ALDH1A1KDM4EPIK3CDPIK3CAPIK3CB
SCHEMBL10878540 0.76 ALDH1A1 (0.49) ALDH1A1KDM4EUSP2F11IMPDH2
SCHEMBL29368700 0.75 PDGFRB (0.51) ALDH1A1KDM4ECYP17A1PIK3CACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed