SCHEMBL9215557

SCHEMBL9215557

COc1ccc(-c2cccnc2)cc1C#N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.55
BACE1 P56817 1/20 0.55
BACE2 Q9Y5Z0 1/20 0.55
CYP11B2 P19099 6/20 0.54
CYP11B1 P15538 4/20 0.54
CYP19A1 P11511 4/20 0.54
KDM4E B2RXH2 3/20 0.53
MAPK1 P28482 1/20 0.53
HSD17B10 Q99714 1/20 0.53
CYP17A1 P05093 3/20 0.52
MKNK1 Q9BUB5 1/20 0.52
MKNK2 Q9HBH9 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 2/20 0.50
NPC1 O15118 2/20 0.48
RAB9A P51151 1/20 0.48
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
STK10 O94804 1/20 0.47
SLK Q9H2G2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025473 0.95 CTSD (0.52) CTSDBACE1BACE2CYP11B2CYP11B1
SCHEMBL10027761 0.82 STK10 (0.48) CTSDBACE1BACE2CYP11B2CYP11B1
SCHEMBL9218755 0.81 ALDH1A1 (0.53) CYP11B2CYP11B1KDM4ECYP17A1ALDH1A1
SCHEMBL29123961 0.81 MAOB (0.57) KDM4EALDH1A1USP2
SCHEMBL30196133 0.81 KDM4E (0.70) CYP11B2CYP11B1CYP19A1KDM4EMAPK1
SCHEMBL11342031 0.81 KDM4E (0.70) CYP11B2CYP11B1CYP19A1KDM4EMAPK1
Hydrochloric Acid SCHEMBL11336399 0.80 KDM4E (0.68) CYP11B2CYP11B1CYP19A1KDM4EMAPK1
SCHEMBL7279694 0.79 PDGFRB (0.51) CYP11B2CYP11B1CYP19A1KDM4ECYP17A1
SCHEMBL1911847 0.78 NPC1 (0.65) CTSDBACE1BACE2CYP11B2CYP11B1
SCHEMBL6439562 0.77 CYP11B2 (0.56) CYP11B2CYP11B1CYP19A1KDM4ECYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed