SCHEMBL9220154

SCHEMBL9220154

CCOC(=O)CNS(=O)(=O)c1c(N)cc(Cl)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
NR3C1 P04150 4/20 0.40
NR3C2 P08235 4/20 0.40
CYP3A4 P08684 2/20 0.40
PGR P06401 2/20 0.40
ABCB1 P08183 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 2/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 2/20 0.36
TP53 P04637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3489281 0.79 NR3C1 (0.46) ALDH1A1NR3C1NR3C2CYP3A4PGR
SCHEMBL3490788 0.76 CA1 (0.45) ALDH1A1NR3C1NR3C2CYP3A4PGR
SCHEMBL15420133 0.75 ABCB1 (0.47) ALDH1A1ABCB1TDP1GAASMN1; SMN2
SCHEMBL3490280 0.74 NR3C1 (0.42) ALDH1A1NR3C1NR3C2CYP3A4PGR
SCHEMBL3489059 0.72 CYP3A4 (0.47) NR3C1NR3C2CYP3A4PGRTDP1
SCHEMBL9220640 0.72 NR3C1 (0.42) ALDH1A1NR3C1NR3C2CYP3A4PGR
SCHEMBL3490267 0.72 CYP3A4 (0.47) NR3C1NR3C2CYP3A4PGRTDP1
SCHEMBL3821657 0.72 THRB (0.41) ALDH1A1LMNAGAASMN1; SMN2PKM
SCHEMBL3488631 0.71 KMT2A (0.52) ALDH1A1NR3C1NR3C2CYP3A4PGR
SCHEMBL3489898 0.71 NR3C1 (0.44) NR3C1NR3C2CYP3A4PGRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636124-A1 3,4-DIHYDRO-2H-1,2,4-BENZOTHIADIAZINE-1,1-DIOXIDE-3-CARBOXYLIC ACID DERIVATIVES, PREPARATION THEREOF AND DRUGS CONTAINING SAME Aventis Pharma S.A. (FR) 1995-02-01 EP disclosed
WO-1993021170-A1 3,4-DIHYDRO-2H-1,2,4-BENZOTHIADIAZINE-1,1-DIOXIDE-3-CARBOXYLIC ACID DERIVATIVES, PREPARATION THEREOF AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1993-10-28 WO disclosed