SCHEMBL9220486

SCHEMBL9220486

CNC(=S)NNC(=O)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.67
ALDH1A1 P00352 5/20 0.66
GAA P10253 3/20 0.66
NPC1 O15118 3/20 0.66
SMN1; SMN2 Q16637 1/20 0.66
CCR6 P51684 1/20 0.63
POLB P06746 2/20 0.62
LMNA P02545 1/20 0.62
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
KDM4E B2RXH2 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11298577 0.88 RAB9A (0.75) RAB9AALDH1A1GAANPC1SMN1; SMN2
SCHEMBL11414330 0.83 GAA (0.70) RAB9AALDH1A1GAASMN1; SMN2CCR6
SCHEMBL2680169 0.82 ALDH1A1 (0.66) RAB9AALDH1A1GAANPC1SMN1; SMN2
SCHEMBL11599578 0.82 KMT2A (0.86) RAB9AALDH1A1GAANPC1SMN1; SMN2
SCHEMBL2477798 0.81 GAA (0.69) RAB9AALDH1A1GAASMN1; SMN2POLB
SCHEMBL400890 0.81 RAB9A (0.77) RAB9AALDH1A1GAANPC1SMN1; SMN2
SCHEMBL8719394 0.81 RAB9A (0.66) RAB9AALDH1A1GAANPC1SMN1; SMN2
SCHEMBL21978380 0.81 ALDH1A1 (0.63) RAB9AALDH1A1GAANPC1SMN1; SMN2
SCHEMBL31558731 0.80 KMT2A (0.72) RAB9AALDH1A1GAANPC1SMN1; SMN2
SCHEMBL14045090 0.80 RAB9A (0.59) RAB9AALDH1A1GAANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0495226-B1 3-Aryl-5-alkylthio-4H-1,2,4-triazoles for treatment of hyperreflexia due to spinal trauma MERRELL DOW PHARMA (US) 1995-10-11 EP disclosed
US-5260450-A Anticonvulsants MERRELL DOW PHARMACEUTICALS INC. (US) 1993-11-09 US disclosed
US-5158968-A 3-aryl-5-alkylthio-4H-1,2,4-traizoles for treatment of hyperreflexia due to spinal trauma MERRELL DOW PHARMACEUTICALS INC. (US) 1992-10-27 US disclosed
US-5143933-A Anticonvulsants MERRELL DOW PHARMACEUTICALS INC. (US) 1992-09-01 US disclosed
EP-0495226-A2 3-Aryl-5-alkylthio-4H-1,2,4-triazoles for treatment of hyperreflexia due to spinal trauma MERRELL DOW PHARMACEUTICALS INC. (US) 1992-07-22 EP disclosed
WO-1989006125-A1 4-ARALKYL-5-SUBSTITUTED-1,2,4-TRIAZOLE-5-THIOLS SMITHKLINE BECKMAN CORPORATION (US) 1989-07-13 WO disclosed
EP-0323737-A1 4-Aralkyl-5-substituted-1,2,4-triazole-5-thiols SMITHKLINE BEECHAM CORPORATION (US) 1989-07-12 EP disclosed