SCHEMBL9220566

SCHEMBL9220566

O=C(NCCO)c1ccc(OCC2(O)CCNCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.48
POLB P06746 2/20 0.44
NPC1 O15118 7/20 0.44
RAB9A P51151 4/20 0.44
SMYD3 Q9H7B4 1/20 0.42
SPHK2 Q9NRA0 1/20 0.42
SPHK1 Q9NYA1 1/20 0.42
ALDH1A1 P00352 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GLA P06280 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 1/20 0.39
NEK1 Q96PY6 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2341524 0.79 MAPT (0.54) POLBNPC1RAB9AMEN1KMT2A
SCHEMBL6284254 0.79 PARP10 (0.49) ALDH1A1KMT2ACA1CA2
SCHEMBL9212770 0.78 CHRM4 (0.51) SPHK2SPHK1SMN1; SMN2
SCHEMBL9483149 0.74 MEN1 (0.40) MMP13POLBNPC1RAB9AMEN1
SCHEMBL9211504 0.74 TDP1 (0.46) ALDH1A1MEN1KMT2AL3MBTL1SMN1; SMN2
SCHEMBL9215011 0.74 ITGB3 (0.57) NPC1
SCHEMBL10345075 0.72 DRD2 (0.50) MMP13NPC1RAB9AALDH1A1MEN1
SCHEMBL5238412 0.72 SSTR5 (0.39)
SCHEMBL620074 0.71 POLB (0.66) MMP13POLBSPHK2SPHK1ALDH1A1
SCHEMBL6285915 0.69 MAPT (0.50) ALDH1A1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0320032-B1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA NV (BE) 1995-01-18 EP disclosed
US-5231184-A Viricide intermediate JANSSEN PHARMACEUTICA N.V. (BE) 1993-07-27 US disclosed
US-5106973-A Viricide intermediates JANSSEN PHARMACEUTICA N.V. (BE) 1992-04-21 US disclosed
US-4992433-A Viricides JANSSEN PHARMACEUTICA N.V. (BE) 1991-02-12 US disclosed
EP-0320032-A1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1989-06-14 EP disclosed