SCHEMBL9211504

SCHEMBL9211504

CCOC(=O)c1ccc(OCC2(O)CCNCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
ESR1 P03372 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
ESR2 Q92731 1/20 0.45
CA14 Q9ULX7 1/20 0.45
STS P08842 1/20 0.45
MAPT P10636 3/20 0.44
LMNA P02545 4/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAOA P21397 1/20 0.44
KCNH2 Q12809 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
ALDH1A1 P00352 2/20 0.43
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2341524 0.86 MAPT (0.54) TDP1L3MBTL1CA1CA2MAPT
SCHEMBL6284254 0.81 PARP10 (0.49) CA1CA2ALDH1A1KMT2A
SCHEMBL9209237 0.77 LMNA (0.55) L3MBTL1LMNACYP3A4ALDH1A1KMT2A
SCHEMBL5155302 0.75 LMNA (0.43) TDP1L3MBTL1CA12CA1CA2
SCHEMBL76052 0.75 ALDH1A1 (0.66) TDP1L3MBTL1CA12CA1CA2
SCHEMBL9220566 0.74 MMP13 (0.48) L3MBTL1CA12CA1CA2CA9
SCHEMBL5238412 0.74 SSTR5 (0.39) LMNA
SCHEMBL10345075 0.74 DRD2 (0.50) ALDH1A1KMT2AMEN1NPSR1
SCHEMBL2343249 0.74 OPRM1 (0.41) MAOAALDH1A1OPRM1
SCHEMBL6701399 0.73 TDP1 (0.74) TDP1L3MBTL1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0320032-B1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA NV (BE) 1995-01-18 EP disclosed
US-5231184-A Viricide intermediate JANSSEN PHARMACEUTICA N.V. (BE) 1993-07-27 US disclosed
US-5106973-A Viricide intermediates JANSSEN PHARMACEUTICA N.V. (BE) 1992-04-21 US disclosed
US-4992433-A Viricides JANSSEN PHARMACEUTICA N.V. (BE) 1991-02-12 US disclosed
EP-0320032-A1 Pyridizinamine derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1989-06-14 EP disclosed