SCHEMBL9225707

SCHEMBL9225707

Cc1cccc(C)c1NC(=O)N(Cc1ccc2c(c1)Cc1ccccc1-2)C1CCCCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
LMNA P02545 1/20 0.43
THRB P10828 1/20 0.42
NPSR1 Q6W5P4 2/20 0.42
TSHR P16473 1/20 0.42
ATM Q13315 1/20 0.42
TP53 P04637 3/20 0.41
MAPT P10636 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
LTB4R2 Q9NPC1 1/20 0.39
CYP1A2 P05177 1/20 0.39
ADRA2A P08913 1/20 0.39
MAOA P21397 1/20 0.39
SLC6A2 P23975 1/20 0.39
HTR2C P28335 1/20 0.39
SLC6A4 P31645 1/20 0.39
HTR2B P41595 1/20 0.39
EPHX1 P07099 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9227832 0.93 NPSR1 (0.45) ALDH1A1LMNATHRBNPSR1TSHR
SCHEMBL4106190 0.93 NPSR1 (0.45) ALDH1A1LMNATHRBNPSR1TSHR
SCHEMBL29427715 0.93 NPSR1 (0.45) ALDH1A1LMNATHRBNPSR1TSHR
SCHEMBL9219992 0.89 SMN1; SMN2 (0.45) ALDH1A1LMNANPSR1TSHRATM
SCHEMBL9225885 0.88 UBE2M (0.51) ALDH1A1NPSR1TSHRATMTP53
SCHEMBL9222967 0.85 ALDH1A1 (0.41) ALDH1A1NPSR1TSHRATMTP53
SCHEMBL9218431 0.85 ALDH1A1 (0.41) ALDH1A1NPSR1TSHRATMTP53
SCHEMBL9537623 0.84 ALDH1A1 (0.42) ALDH1A1LMNATHRBNPSR1TSHR
SCHEMBL9222936 0.84 NPSR1 (0.43) ALDH1A1LMNANPSR1TSHRATM
SCHEMBL9220959 0.83 GAA (0.50) ALDH1A1LMNATHRBNPSR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420348-A Enzyme inhibitors YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0447116-B1 Urea derivatives, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMA CO LTD (JP) 1994-12-14 EP disclosed
US-5258405-A Acetyl coenzyme A cholesterol acetyltransferase inhibitors for cardiovascular disorders and atherosclerosis and antilipemic agents YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1993-11-02 US disclosed
EP-0447116-A1 Urea derivatives, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-09-18 EP disclosed