SCHEMBL9229883

SCHEMBL9229883

Cc1cc(=O)oc2c(N3CCNCC3)cccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 2/20 0.52
ADRB1 P08588 3/20 0.50
KMT2A Q03164 1/20 0.47
HTR7 P34969 3/20 0.47
HTR6 P50406 2/20 0.47
NCF1 P14598 2/20 0.47
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
CYP1A2 P05177 1/20 0.47
HTR1A P08908 1/20 0.47
CYP2D6 P10635 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
HTR1D P28221 1/20 0.47
HTR1B P28222 1/20 0.47
HTR2A P28223 1/20 0.47
MTOR P42345 1/20 0.47
HTR3A P46098 1/20 0.47
HTR5A P47898 1/20 0.47
HTR3D Q70Z44 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9229213 0.78 KMT2A (0.57) KMT2ANCF1HTR1AHTR2AALDH1A1
SCHEMBL9229904 0.77 ADRB1 (0.51) ADRB1HTR7HTR6NCF1HTR3E
Hydrochloric Acid SCHEMBL9229290 0.76 ADRB1 (0.50) ADRB1HTR7HTR6NCF1HTR3E
Batoprazine SCHEMBL766463 0.76 HTR5A (0.53) ADRB1HTR7HTR6NCF1HTR3E
Formamide SCHEMBL27876319 0.74 ADRB1 (0.48) ADRB1HTR7HTR6NCF1HTR3E
SCHEMBL5904424 0.72 KMT2A (0.64) PRKDCKMT2ACYP1A2TSHRHSD17B10
SCHEMBL30940063 0.72 KMT2A (0.64) PRKDCKMT2ACYP1A2TSHRHSD17B10
SCHEMBL5203993 0.71 PRKDC (0.73) PRKDCHTR7HTR6NCF1HTR3E
SCHEMBL1443282 0.71 DRD2 (0.56) ADRB1HTR6HTR1AHTR2A
SCHEMBL16156549 0.71 ADRB1 (0.69) ADRB1HTR7HTR6NCF1HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1105360-A 1-[2H-1-benzopyran-2-one-8yl]-piperazin derivative DUPHAR INT RES (NL) 1995-07-19 CN disclosed
EP-0650964-A1 1 2H-1-benzopyran-2-one-8-yl -piperazine derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1995-05-03 EP disclosed