SCHEMBL9232256

SCHEMBL9232256

Cc1c(OC(=O)O)[nH]c2ccc(F)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
KIF11 P52732 1/20 0.43
KDM4E B2RXH2 5/20 0.42
MAPT P10636 1/20 0.42
ALDH1A1 P00352 4/20 0.42
HPGD P15428 3/20 0.42
THRB P10828 1/20 0.42
MAP2 P11137 1/20 0.42
FEN1 P39748 1/20 0.41
GABRA1 P14867 2/20 0.40
GABRG2 P18507 2/20 0.40
GABRB3 P28472 2/20 0.40
GABRA5 P31644 2/20 0.40
GABRA3 P34903 2/20 0.40
GABRA2 P47869 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRL1 P41146 1/20 0.40
GABRA4 P48169 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27908888 0.89 KEAP1 (0.47) KEAP1NFE2L2KIF11KDM4EMAPT
SCHEMBL9231630 0.81 DRD2 (0.44) KEAP1NFE2L2KDM4EMAP2GABRA1
SCHEMBL2730323 0.78 ALDH1A1 (0.59) KEAP1NFE2L2KIF11KDM4EMAPT
SCHEMBL6583063 0.73 TUBB4A (0.51) KEAP1NFE2L2KDM4EALDH1A1HPGD
SCHEMBL15101537 0.73 TSHR (0.52) KEAP1NFE2L2KIF11KDM4EMAPT
SCHEMBL7371534 0.72 KDM4E (0.50) KEAP1NFE2L2KDM4EMAPTALDH1A1
SCHEMBL2730512 0.72 MAP2 (0.61) KEAP1NFE2L2KIF11KDM4EMAPT
SCHEMBL14255879 0.72 KMT2A (0.55) KEAP1NFE2L2KIF11KDM4EMAPT
SCHEMBL30356394 0.71 MAPT (0.55) KEAP1NFE2L2KIF11KDM4EMAPT
SCHEMBL10067335 0.71 MAPT (0.55) KEAP1NFE2L2KIF11KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655440-A2 1-Aminoethylindoles F. HOFFMANN-LA ROCHE AG (CH) 1995-05-31 EP disclosed