SCHEMBL9244182

SCHEMBL9244182

Cn1c(OC(=O)O)c(S(=O)(=O)c2ccccc2)c2cc(Cl)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.44
PTGDR2 Q9Y5Y4 3/20 0.43
AKR1B1 P15121 1/20 0.42
HTR6 P50406 2/20 0.40
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40
TUBA1A Q71U36 1/20 0.40
TUBA1C Q9BQE3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9238450 0.90 EGFR (0.44) EGFRPTGDR2AKR1B1HTR6MAPT
SCHEMBL8689826 0.82 ACLY (0.48) EGFRPTGDR2AKR1B1HTR6MAPT
SCHEMBL8687705 0.81 KDM4E (0.53) EGFRPTGDR2AKR1B1MAPTNPSR1
SCHEMBL9241871 0.77 EGFR (0.43) EGFRMAPTLMNAHTTKDM4E
SCHEMBL9236400 0.77 ACLY (0.47) EGFRMAPTACLYKDM4EKMT2A
SCHEMBL11613647 0.77 EGFR (0.45) EGFRPTGDR2HTR6MAPTLMNA
SCHEMBL9240535 0.76 EGFR (0.42) EGFRMAPTLMNAKDM4ETSHR
SCHEMBL9240069 0.72 TUBB4A (0.50) MAPTNPSR1TUBB4ATUBBTUBA3C
SCHEMBL19547602 0.69 ENPP2 (0.45) PTGDR2AKR1B1LMNANPSR1KDM4E
SCHEMBL9266263 0.68 OXER1 (0.64)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639573-A1 Benzocondensed five membered heterocycles, process of their preparation, their use as drug, as diagnostic means and pharmaceuticals containing it HOECHST AKTIENGESELLSCHAFT (DE) 1995-02-22 EP disclosed