SCHEMBL8687705

SCHEMBL8687705

COC(=O)c1c(S(=O)(=O)c2ccccc2)c2cc(Cl)ccc2n1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 1/20 0.53
HPGD P15428 1/20 0.53
HSD17B10 Q99714 1/20 0.53
TUBB4A P04350 1/20 0.45
TUBB P07437 1/20 0.45
TUBA3C P0DPH7 1/20 0.45
TUBA1B P68363 1/20 0.45
TUBA4A P68366 1/20 0.45
TUBB4B P68371 1/20 0.45
TUBB3 Q13509 1/20 0.45
TUBB2A Q13885 1/20 0.45
TUBB8 Q3ZCM7 1/20 0.45
TUBA3E Q6PEY2 1/20 0.45
TUBA1A Q71U36 1/20 0.45
TUBA1C Q9BQE3 1/20 0.45
TUBB6 Q9BUF5 1/20 0.45
TUBB2B Q9BVA1 1/20 0.45
TUBB1 Q9H4B7 1/20 0.45
EGFR P00533 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689826 0.88 ACLY (0.48) KDM4EHSD17B10EGFRPTGDR2MAPT
SCHEMBL9238450 0.83 EGFR (0.44) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL9244182 0.81 EGFR (0.44) KDM4ETUBB4ATUBBTUBA3CTUBA1B
SCHEMBL22022202 0.78 PLA2G2A (0.52) KDM4EALDH1A1HPGDHSD17B10EGFR
SCHEMBL21478268 0.76 PABPC1 (0.46) KDM4EALDH1A1HPGDHSD17B10EGFR
SCHEMBL24482986 0.75 ALDH1A1 (0.43) KDM4EALDH1A1HPGDHSD17B10EGFR
SCHEMBL11613647 0.75 EGFR (0.45) KDM4EALDH1A1HPGDEGFRPTGDR2
SCHEMBL5234885 0.71 SMN1; SMN2 (0.52) KDM4EALDH1A1HPGDHSD17B10EGFR
SCHEMBL11532944 0.71 ALDH1A1 (0.51) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL22003908 0.70 ACLY (0.78) PTGDR2MAPK8MAPTMAPK9ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852046-A Benzo-fused heterocyclic compounds having a 5-membered ring processes for their preparation their use as medicaments their use as diagnostic agents and medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1998-12-22 US disclosed