SCHEMBL9253948

SCHEMBL9253948

C=CCCCc1cnc(-c2ccc(F)c(F)c2)nc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 1/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
CYP17A1 P05093 1/20 0.35
NOTUM Q6P988 1/20 0.33
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
GPR68 Q15743 1/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
DYRK1B Q9Y463 1/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HSD17B10 Q99714 2/20 0.32
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32
PKM P14618 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9251920 0.94 CYP11B1 (0.39) RARBCYP11B1CYP11B2CYP17A1NOTUM
SCHEMBL9249705 0.91 CYP11B1 (0.36) RARBCYP11B1CYP11B2CYP17A1NOTUM
SCHEMBL9252364 0.86 CYP11B1 (0.41) RARBCYP11B1CYP11B2CYP17A1GRIN1
SCHEMBL9253679 0.84 RARB (0.40) RARBCYP11B1CYP11B2GRIN2BRAB9A
SCHEMBL9252022 0.82 RARB (0.40) RARBGRIN2BRAB9ASMN1; SMN2HSD17B10
SCHEMBL9353374 0.82 CYP11B1 (0.38) CYP11B1CYP11B2CYP17A1NOTUMGRIN1
SCHEMBL10515024 0.81 CYP11B2 (0.43) CYP11B1CYP11B2
SCHEMBL9253788 0.81 RARB (0.40) RARBRAB9ASMN1; SMN2HSD17B10NPC1
SCHEMBL10728895 0.81 RARB (0.50) RARBPDGFRBPDGFRARAB9ASMN1; SMN2
SCHEMBL7516234 0.79 RARB (0.56) RARBRAB9ASMN1; SMN2HSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5454974-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1995-10-03 US disclosed
US-5302317-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1994-04-12 US disclosed
EP-0315014-B1 Halogenated benzene derivatives HOFFMANN LA ROCHE (CH) 1994-01-12 EP disclosed
US-5230826-A HALOBENZENE LIQUID CRYSTALS HOFFMANN-LA ROCHE INC. (US) 1993-07-27 US disclosed
EP-0315014-A2 Halogenated benzene derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed