SCHEMBL9250252

SCHEMBL9250252

COc1cc2ccc(Br)cc2c(C(=O)O)c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
LMNA P02545 3/20 0.44
POLB P06746 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
RXFP1 Q9HBX9 5/20 0.43
PRNP P04156 2/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
PPARG P37231 1/20 0.43
NR2E3 Q9Y5X4 1/20 0.43
NCOR2 Q9Y618 1/20 0.43
PTGFR P43088 2/20 0.43
TP53 P04637 1/20 0.43
HSD17B10 Q99714 1/20 0.42
DHODH Q02127 1/20 0.42
CA12 O43570 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24150723 0.83 CA12 (0.49) ALDH1A1HTTL3MBTL1SMN1; SMN2LMNA
SCHEMBL9736420 0.82 NCEH1 (0.46) ALDH1A1HTTL3MBTL1SMN1; SMN2LMNA
SCHEMBL11507377 0.79 POLB (0.56) ALDH1A1L3MBTL1SMN1; SMN2LMNAPOLB
SCHEMBL27619794 0.76 CA12 (0.50) ALDH1A1HTTL3MBTL1SMN1; SMN2LMNA
SCHEMBL19328740 0.75 PTGFR (0.62) ALDH1A1HTTMEN1KMT2ARXFP1
SCHEMBL9039455 0.73 CYP3A4 (0.55) ALDH1A1HTTL3MBTL1LMNAPOLB
SCHEMBL18481324 0.73 ALDH1A1 (0.50) ALDH1A1HTTSMN1; SMN2MEN1KMT2A
SCHEMBL358180 0.72 KDM4E (0.70) ALDH1A1LMNAPOLBMEN1KMT2A
SCHEMBL8346118 0.71 ALDH1A1 (0.41) ALDH1A1HTTL3MBTL1SMN1; SMN2LMNA
SCHEMBL6828042 0.71 MEN1 (0.48) ALDH1A1L3MBTL1POLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5426189-A Dopamine receptor ligands and imaging agents THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1995-06-20 US disclosed
US-5334728-A Dopamine receptor ligands and imaging agents THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1994-08-02 US disclosed
US-5186921-A 3-methoxy-n(1-ethyl-2-pyrrolidinyl)methyl)naphthyl-2-carboxy amide compounds for imaging human brains; good retention stability TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1993-02-16 US disclosed
US-5122361-A 2-Pyrrolidinylmethylcarboxamido-2,3-dihydrobenzofuran type compounds TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1992-06-16 US disclosed
EP-0393838-A1 Dopamine receptor ligands and imaging agents THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1990-10-24 EP disclosed