SCHEMBL9251106

SCHEMBL9251106

CCN(Cc1c(C(=O)O)[nH]c2ccc(C)cc12)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.51
ALDH1A1 P00352 5/20 0.51
HPGD P15428 3/20 0.49
MAPT P10636 3/20 0.49
HSD17B10 Q99714 2/20 0.49
USP2 O75604 1/20 0.49
MAPK1 P28482 1/20 0.49
CASP7 P55210 1/20 0.49
CNR1 P21554 1/20 0.47
OPRM1 P35372 3/20 0.45
EGFR P00533 1/20 0.43
CDK2 P24941 1/20 0.43
ACHE P22303 1/20 0.43
SIGMAR1 Q99720 3/20 0.43
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
HTT P42858 3/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9260626 0.93 KDM4E (0.51) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL9255557 0.91 ALDH1A1 (0.50) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL27350858 0.91 OPRM1 (0.48) OPRM1EGFRCDK2SIGMAR1KMT2A
SCHEMBL27439205 0.84 OPRM1 (0.48) OPRM1SIGMAR1KMT2ACHRM3OPRD1
SCHEMBL9260006 0.84 CNR1 (0.53) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL9251803 0.83 ACHE (0.50) KDM4EALDH1A1HPGDOPRM1ACHE
SCHEMBL9264547 0.80 SLC6A2 (0.47) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL9254627 0.80 KDM4E (0.51) KDM4EALDH1A1OPRM1ACHESIGMAR1
SCHEMBL9261885 0.78 KDM4E (0.51) KDM4EALDH1A1OPRM1ACHESIGMAR1
SCHEMBL9251113 0.78 ACHE (0.54) KDM4EALDH1A1HPGDMAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428043-A Tricyclic-cyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1995-06-27 US disclosed
EP-0441517-A2 Tricyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1991-08-14 EP disclosed