SCHEMBL9251384

SCHEMBL9251384

CC(C)C(NC(=O)C(CC(=O)O)NC(=O)c1ccc2c(c1)nc(-c1ccc(C(=N)N)cc1)n2C)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.49
HDAC8 Q9BY41 3/20 0.49
HDAC6 Q9UBN7 3/20 0.49
HDAC3 O15379 2/20 0.48
HDAC2 Q92769 2/20 0.48
NAMPT P43490 1/20 0.43
PTGER4 P35408 2/20 0.39
F2 P00734 6/20 0.39
PRSS1 P07477 5/20 0.39
TMPRSS15 P98073 4/20 0.39
JAK2 O60674 2/20 0.38
JAK1 P23458 2/20 0.38
TYK2 P29597 2/20 0.38
JAK3 P52333 2/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
SLC22A2 O15244 1/20 0.37
F10 P00742 1/20 0.37
PLG P00747 1/20 0.37
PLAT P00750 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9248512 0.90 HDAC1 (0.56) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9250758 0.86 HDAC6 (0.52) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9252732 0.85 HDAC1 (0.46) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9252518 0.83 PRSS1 (0.46) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9251560 0.80 ITGB3 (0.47) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9252202 0.78 HDAC6 (0.55) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9249572 0.78 ITGB3 (0.56) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9249490 0.78 HDAC1 (0.56) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9251773 0.75 HDAC1 (0.50) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9255124 0.75 HDAC1 (0.50) HDAC1HDAC8HDAC6HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed