SCHEMBL9251560

SCHEMBL9251560

COc1ccc(CCNC(=O)C(CC(=O)O)NC(=O)c2ccc3c(c2)nc(-c2ccc(C(=N)N)cc2)n3C)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.47
ITGA2B P08514 5/20 0.47
HDAC1 Q13547 3/20 0.44
HDAC8 Q9BY41 3/20 0.44
HDAC6 Q9UBN7 3/20 0.44
HDAC3 O15379 2/20 0.44
HDAC2 Q92769 2/20 0.44
PRSS1 P07477 2/20 0.43
TMPRSS15 P98073 2/20 0.43
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ENPP2 Q13822 1/20 0.41
THRB P10828 1/20 0.40
F2 P00734 2/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9252518 0.88 PRSS1 (0.46) ITGB3ITGA2BHDAC1HDAC8HDAC6
SCHEMBL9248512 0.82 HDAC1 (0.56) ITGB3ITGA2BHDAC1HDAC8HDAC6
SCHEMBL9252697 0.82 HDAC6 (0.42) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9251384 0.80 HDAC1 (0.49) ITGB3ITGA2BHDAC1HDAC8HDAC6
SCHEMBL9252732 0.80 HDAC1 (0.46) ITGB3ITGA2BHDAC1HDAC8HDAC6
SCHEMBL9250758 0.79 HDAC6 (0.52) ITGB3ITGA2BHDAC1HDAC8HDAC6
Hydrochloric Acid SCHEMBL8886078 0.79 ITGB3 (0.59) ITGB3ITGA2BPRSS1TMPRSS15F2
SCHEMBL9252703 0.79 ENPP2 (0.39) ITGB3ITGA2BHDAC6PRSS1TMPRSS15
Hydrochloric Acid SCHEMBL8885572 0.78 ITGB3 (0.56) ITGB3ITGA2BPRSS1TMPRSS15NPC1
SCHEMBL9249490 0.76 HDAC1 (0.56) ITGB3ITGA2BHDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed