SCHEMBL9251891

SCHEMBL9251891

C#CC[CH]c1cccc(C#N)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 3/20 0.45
GRIN2D O15399 2/20 0.44
GRIN3B O60391 2/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
GRIN2B Q13224 2/20 0.44
GRIN2C Q14957 2/20 0.44
GRIN3A Q8TCU5 2/20 0.44
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
P4HB P07237 8/20 0.40
ENPP2 Q13822 1/20 0.38
DRD2 P14416 1/20 0.37
GSK3B P49841 1/20 0.37
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16619152 0.79 PDCD1 (0.50) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL27336648 0.78 GRIN2D (0.50) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7331821 0.76 PDCD1 (0.48) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3208694 0.76 FBP1 (0.49) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8668592 0.75 FBP1 (0.45) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL29463498 0.75 FBP1 (0.56) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3216977 0.75 FBP1 (0.51) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL67236 0.75 FBP1 (0.56) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL2774364 0.74 FBP1 (0.65) FBP1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL1687910 0.74 FBP1 (0.65) FBP1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5395838-A Aromatic aminomethyl substitutes compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-03-07 US disclosed
US-5252573-A Quinazoline derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-12 US disclosed
US-5089499-A Anticarcinogenic agents; thymidylate synthetase inhibitors; antiallergens; psoriasis IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-02-18 US disclosed