SCHEMBL9252129

SCHEMBL9252129

CNc1cc2c(cc1C(=O)NCCC(=O)OC)nc(-c1ccc(C#N)cc1)n2C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 2/20 0.41
EGLN1 Q9GZT9 2/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
ITK Q08881 3/20 0.38
EGLN2 Q96KS0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
TRPA1 O75762 1/20 0.36
TNF P01375 1/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
BRD4 O60885 1/20 0.36
PTGER4 P35408 2/20 0.35
ADORA2A P29274 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC2 Q92769 1/20 0.35
KDM1A O60341 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9248585 0.85 EGLN1 (0.37) IRAK4EGLN1JAK2JAK1TYK2
SCHEMBL9255968 0.84 HDAC1 (0.51) EGLN1JAK2JAK1TYK2JAK3
Acetic Acid SCHEMBL9256132 0.82 CHEK2 (0.39) KDM5BHDAC1HDAC8HDAC6PTGER4
SCHEMBL9255248 0.81 IRAK4 (0.37) IRAK4EGLN1JAK2JAK1TYK2
SCHEMBL9256202 0.78 JAK2 (0.55) JAK2JAK1TYK2JAK3ITK
SCHEMBL9250822 0.77 ADORA2A (0.46) IRAK4EGLN1JAK2JAK1TYK2
SCHEMBL9249905 0.77 CHEK2 (0.39) KDM5BHDAC1HDAC8HDAC6HDAC3
SCHEMBL9251414 0.76 CHEK2 (0.38) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9253691 0.76 JAK2 (0.60) JAK2JAK1TYK2JAK3ITK
SCHEMBL9254520 0.75 ITGB3 (0.44) HDAC1HDAC8HDAC6HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed