SCHEMBL9253096

SCHEMBL9253096

COC(=O)NC(=N)c1ccc(-c2cn(C)c(-c3ccc(CCC(=O)OCCc4ccccc4)cc3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.40
ALOX5 P09917 1/20 0.40
APP P05067 1/20 0.40
MAPT P10636 1/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
KDM4E B2RXH2 2/20 0.36
HPGD P15428 2/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 3/20 0.36
NAMPT P43490 2/20 0.35
ROCK2 O75116 1/20 0.34
THRB P10828 1/20 0.34
VCP P55072 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257104 0.89 HRH3 (0.39) TDP1MAPTHPGDGAAALDH1A1
SCHEMBL9288922 0.87 TDP1 (0.43) TDP1ALOX5APPMAPTKDM4E
SCHEMBL9255728 0.86 KDM4E (0.37) TDP1KDM4EHPGDMEN1GAA
SCHEMBL9247334 0.85 PTGDR2 (0.40)
SCHEMBL9255100 0.84 KDM4E (0.36) PPARGPPARAKDM4EHPGDMEN1
SCHEMBL9256151 0.83 HPGD (0.35) MAPTHPGDNAMPT
SCHEMBL9257842 0.82 HRH3 (0.34) TDP1MAPTHPGDGAAALDH1A1
SCHEMBL9254248 0.82 CASP1 (0.35) KDM4EHPGDGAAALDH1A1
SCHEMBL9256883 0.81 KDM4E (0.36) MAPTKDM4EHPGDMEN1GAA
SCHEMBL9250731 0.80 HRH3 (0.34) TDP1MAPTHPGDGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed